1084889-77-9Relevant articles and documents
Convergent synthesis of dihydroquinolones from o-aminoarylboronates
Horn, Joachim,Li, Ho Yin,Marsden, Stephen P.,Nelson, Adam,Shearer, Rachel J.,Campbell, Amanda J.,House, David,Weingarten, Gordon G.
experimental part, p. 9002 - 9007 (2009/12/22)
An efficient and convergent one-step synthesis of substituted dihydroquinolin-2-ones from α,β-unsaturated esters and aminoaryl pinacolboronates under rhodium catalysis is reported. The reaction is easily applicable in parallel synthesis format and provide