1097200-61-7Relevant articles and documents
Enol phosphinates and phosphonates: Practical electrophiles for cross-coupling strategies
Steel, Patrick G.,Woods, Tom M.
experimental part, p. 3897 - 3904 (2010/03/24)
Enol phosphinates and phosphonates can be readily prepared from simple lactams in high yields and are both stable and storable. Both these substrates can be employed successfully in homogeneous Suzuki-Miyaura and Stille cross-couplings protocols. Additionally, the phosphonate group can be immobilised on a phenol-on-polystyrene resin and utilised in a simple diversity linker strategy in which the coupled product is cleaved from the resin under Suzuki-Miyaura cross-coupling conditions. Georg Thieme Verlag Stuttgart.
