111600-89-6Relevant articles and documents
HETEROCYCLIC COMPOUNDS AND USES THEREOF
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Paragraph 00655; 00659; 00709, (2015/04/22)
Compounds and pharmaceutical compositions that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including PI3 kinase activity, are described herein.
HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF PI3K-GAMMA MEDIATED DISORDERS
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Paragraph 001311; 001315, (2015/11/10)
Compounds and pharmaceutical compositions that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including PI3 kinase activity, are described herein.
p-Substituted Asymmetric Ureas and Medical Uses Thereof
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Paragraph 0253; 0255, (2015/09/28)
Disclosed are compounds, compositions and methods for the prevention and/or treatment of diseases which are pathophysiologically mediated by the ghrelin receptor. The compounds have the general Formula I: or pharmaceutically acceptable salts thereof.
2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS
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Page/Page column 26-27, (2008/12/08)
Anti-viral agents of compounds of Formula (I) : wherein A, Rx, Ry, R2 and R3 are as defined in the specification, processes for their preparation and their use in HCV treatment are provided.
2-Thioethenyl substituted carbapenem derivatives
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Page/Page column 22, (2010/11/25)
[Objective] An objective of the present invention is to provide compounds that are effective against various resistant bacteria which cause current clinical problems, for example, pneumococci including penicillin resistant Streptococcus pneumoneae (PRSP),
INDOLE COMPOUNDS USEFUL AS IMPDH INHIBITORS
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Page column 42-43, (2010/02/04)
Compounds having the Formula (I), are effective as inhibitors of IMPDH enzyme, wherein R3 is alkyl, substituted alkyl, alkoxy, haloalkoxy, or halogen, preferably methoxy, ethoxy, or trifluoromethoxy; and R1, R2, R4, and R5 are as defined in the specificat
Palladium-Catalyzed Reactions of Terminal Acetylenes and Olefins with Halo-1,3-azoles
Sakamoto, Takao,Nagata, Hideo,Kondo, Yoshinori,Shiraiwa, Masafumi,Yamanaka, Hiroshi
, p. 823 - 828 (2007/10/02)
The palladium-catalyzed reactions of 4-bromo- and 5-bromothiazoles, as well as 4-bromo and 5-bromooxazoles with terminal acetylenes gave ethynyl derivatives in 43-89percent yields, whereas the reactions of 2-bromothiazoles and iodo-N-methylimidazoles affo