112225-90-8Relevant academic research and scientific papers
Synthesis and insecticidal activity of chromanone and chromone analogues of diacylhydrazines
Zhao, Pei-Liang,Li, Jing,Yang, Guang-Fu
, p. 1888 - 1895 (2007)
Diacylhydrazine derivatives have been identified as one of the most important insect growth regulators. A variety of diacylhydrazine derivatives were designed and synthesized in recent years due to their unique action mechanism, simple structure, and environmental benign character. This paper describes the molecular design, synthesis, and insecticidal activities of a series of chromanone and chromone analogues of diacylhydrazine derivatives. The preliminary bioassay showed that some of the chromanone analogues exhibited good insecticidal activity against Mythima separata at the dosage of 500 mg L-1. The present work demonstrated that replacement of the chroman ring of ANS-118, a commercial insecticide, with chromanone moiety could result in new compounds with high potent insecticidal activity.
Synthesis and Bioactivities Evaluation of Novel Anthranilic Diamides Containing N-(tert-Butyl)benzohydrazide Moiety as Potent Ryanodine Receptor Activator
Zhou, Yunyun,Wei, Wei,Zhu, Liangliang,Li, Yuxin
supporting information, p. 605 - 610 (2019/05/10)
Anthranilic diamides have been proven to be a class of efficacious and safe insecticides targeting ryanodine receptors (RyRs) during the last decade. In order to develop innovative scaffolds with high insecticidal activity, two series of N-pyridylpyrazole
Diacylhydrazine derivatives as well as preparation method and application thereof
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Paragraph 0057; 0059; 0060, (2019/02/06)
The invention belongs to the field of agricultural insecticides and particularly provides a preparation method and an application of diacylhydrazine insecticides. The compounds improve lipid solubility of original compounds and further have excellent inse
Copper-catalyzed synthesis of substituted indazoles from 2-chloroarenes at low catalyst-loading
Tanimori, Shinji,Kobayashi, Yasuyuki,Iesaki, Yasukazu,Ozaki, Yuka,Kirihata, Mitsunori
experimental part, p. 1381 - 1387 (2012/04/04)
An efficient and convenient access to 1-substituted indazol-3-ones 2 has been achieved throughout the intramolecular C-N bond formations of 2-chloro-benzoic acid-N′-aryl and alkyl-hydrazides employing 0.5 mol% of cuprous (I) iodide and 20 mol% of l-prolin
Synthesis and insecticidal activity of N - Tert -Butyl- N, N ′-diacylhydrazines containing 1,2,3-thiadiazoles
Wang, Huan,Yang, Zhikun,Fan, Zhijin,Wu, Qingjun,Zhang, Youjun,Mi, Na,Wang, Shouxin,Zhang, Zhengcai,Song, Haibin,Liu, Feng
experimental part, p. 628 - 634 (2011/10/02)
N-tert-Butyl-N,N′-diacylhydrazines are nonsteroidal ecdysone agonists used as environmental benign pest regulators. In this paper, two series of new N-tert-butyl-N,N′-diacylhydrazine derivatives containing 1,2,3-thiadiazole were designed and synthesized.
Quantitative structure-activity studies of insect growth regulators: XVI. Substituent effects of dibenzoylhydrazines on the insecticidal activity to Colorado potato beetle Leptinotarsa decemlineata
Nakagawa,Smagghe,Kugimiya,Hattori,Ueno,Tirry,Fujita
, p. 909 - 918 (2007/10/03)
Insecticidal activity against the Colorado potato beetle, Leptinotarsa decemlineata, was measured for a series of substituted N-tert-butyl- dibenzoylhydrazines, in which one of the benzoyl moieties closer to the tert- butyl group was fixed as being 2-chlo
