1123630-10-3Relevant academic research and scientific papers
A practical protocol for three-component, one-pot, stepwise sonogashira-heterocyclization-heck couplings
Madich, Youssef,Denis, J.Gabriel,Ortega, Aitor,Martinez, Claudio,Matrane, Abdellatif,Belachemi, Larbi,De Lera, Angel R.,Alvarez, Rosana,Aurrecoechea, Jose M.
, p. 2009 - 2017 (2013/07/26)
A three-component, one-pot, stepwise Sonogashira-heterocyclization-Heck- coupling process was developed starting from either haloarenecarboxamides, halophenols or haloanilines, terminal alkynes and electron-deficient alkenes. Cyclic imidate-, benzofuran-,
A general synthesis of alkenyl-substituted benzofurans, indoles, and isoquinolones by cascade palladium-catalyzed heterocyclization/oxidative heck coupling
Alvarez, Rosana,Martinez, Claudio,Madich, Youssef,Denis, J. Gabriel,Aurrecoechea, Jose M.,De Lera, Angel R.
supporting information; experimental part, p. 12746 - 12753 (2011/02/21)
Structurally diverse C3-alkenylbenzofurans, C3-alkenylindoles, and C4-alkenylisoquinolones are efficiently prepared by using consecutive Sonogashira and cascade Pd-catalyzed heterocyclization/oxidative Heck couplings from readily available ortho-iodosubst
Palladium-catalyzed sequential oxidative cyclization/coupling of 2-alkynylphenols and alkenes: A direct entry into 3-alkenylbenzofurans
Martinez, Claudio,Alvarez, Rosana,Aurrecoechea, Jose M.
supporting information; experimental part, p. 1083 - 1086 (2009/07/25)
A new Pd-catalyzed tandem intramolecular oxypalladation/Heck-type coupling between 2-alkynylphenols and alkenes is reported, leading to 3-(1-alkenyl)benzofurans. Participating alkenes include those substituted with an electron-withdrawing group (ester, ke
