1132879-15-2Relevant academic research and scientific papers
Novel azoles as potent and selective cannabinoid CB2 receptor agonists
Harnett, Jeremiah J.,Dolo, Christine,Viossat, Isabelle,Auger, Florence,Ferrandis, Eric,Bigg, Dennis,Auguet, Michel,Auvin, Serge,Chabrier, Pierre-E.
, p. 88 - 91 (2015/02/19)
Novel azole compounds were prepared which demonstrated potent hCB2 binding activities with antioxidant activity for a selected compound. These compounds show good selectivity over the hCB1 receptor and are full agonists at the hCB2 receptor.
4-PHENYL-1,3-THIAZOLES AND 4-PHENYL-1,3-OXAZOLES DERIVATIVES AS CANNABINOID RECEPTOR LIGANDS
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Page/Page column 13, (2011/04/18)
The present invention relates to new 4-phenyl-1,3-azole derivatives having the general formula (I) wherein R1, R2, R3, R4, X, A, B, and n are variable, in a racemic form, an enantiomeric form or any combinations thereof. These compounds exhibit affinity f
