1150271-74-1

Usage

Uses

4-Bromomethyl-3-fluorophenylboronic acid, pinacol ester

Upstream product

• 903895-56-7 2-(3-fluoro-4-methylphenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 

Downstream Products

• 1418201-61-2 4-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)benzyl)-2H-benzo[b][1,4]thiazin-3(4H)-one 1,1-dioxide 
• 1418201-60-1 4-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)benzyl)-2H-benzo[b][1,4]thiazin-3(4H)-one-1-oxide 
• 1418201-59-8 4-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)benzyl)-2H-benzo[b][1,4]thiazin-3(4H)-one 

Relevant academic research and scientific papers

A modular approach to catalytic synthesis using a dual-functional linker for Click and Suzuki coupling reactions

The stable benzylazido-boronate ester 1 is presented as an example of a dual-functional linker that allows the synthetically valuable boronate motif to be clicked onto other molecules under mild conditions. The utility of the azido-boronate motif as a modular building block is demonstrated in the rapid synthesis of drug-like structures employing sequential catalytic azide-alkyne cycloaddition and Suzuki coupling reactions.