1152781-66-2Relevant academic research and scientific papers
5-HETEROARYL-PYRIDIN-2-AMINE CONFOUNDS AS NEUROPEPTIDE FF RECEPTOR ANTAGONISTS
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, (2021/02/12)
The present invention relates to novel aminopyridine derivatives of the general formula (I) and pharmaceutical compositions comprising these compounds, as well as their therapeutic use, particularly as neuropeptide FF (NPFF) receptor antagonists, including, e.g., for the treatment or prevention of pain, opioid-induced hyperalgesia, or addiction.
Optimization of TopoIV Potency, ADMET Properties, and hERG Inhibition of 5-Amino-1,3-dioxane-Linked Novel Bacterial Topoisomerase Inhibitors: Identification of a Lead with in Vivo Efficacy against MRSA
Chen, Anna,Cummings, Jason E.,Duncan, Leonard R.,English, Anthony,Koci, Bryan,Li, Linsen,Lindert, Steffen,Lu, Yanran,Mann, Chelsea A.,Mcelroy, Craig A.,Mitton-Fry, Mark J.,Nolan, Sheri,Okumu, Antony,Papa, Jonathan L.,Ratigan, Steven C.,Roth, Brieanna,Seffernick, Justin T.,Slayden, Richard A.,Vibhute, Sandip,Wozniak, Daniel J.,Yalowich, Jack
, p. 15214 - 15249 (2021/10/25)
Novel bacterial topoisomerase inhibitors (NBTIs) are among the most promising new antibiotics in preclinical/clinical development. We previously reported dioxane-linked NBTIs with potent antistaphylococcal activity and reduced hERG inhibition, a key safet
HETEROCYCLIC COMPOUNDS AND USES THEREOF
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, (2019/10/23)
In recognition of the unmet need to develop novel therapeutic agents, the present invention discloses a novel class of heterocycles as dual inhibitors of BRD4 and class I PI3Ks. The compounds claimed herein could be used alone or in combination therapies
5-[(3,3,3-Trifluoro-2-hydroxy-1-arylpropyl)amino]-1-arylquinolin-2-ones, a Process for their Production and their Use as Anti-inflammatory Agents
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Page/Page column 12, (2010/02/17)
The present invention relates to compounds of formula I, processes and intermediates for their production and their use as anti-inflammatory agents.
5-[(3,3,3-Trifluoro-2-hydroxy-1-arylpropyl)amino-1-arylquinolin-2-ones, a process for their production and their use as anti-inflammatory agents
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Page/Page column 20, (2010/03/02)
The present invention relates to compounds of formula I, processes and intermediates for their production and their use as antiinflammatory agents.
5-[(3,3,3-Trifluoro-2-hydroxy-1-arylpropyl)amino]-1H-quinolin-2-ones, A Process for Their Production and Their Use as Anti-inflammatory Agents
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Page/Page column 13, (2009/06/27)
The present invention relates to compounds of formula I, processes for their production and their use as anti-inflammatory agents.
