1160360-15-5Relevant articles and documents
Discovery of fused 5,6-bicyclic heterocycles as γ-secretase modulators
Qin, Jun,Dhondi, Pawan,Huang, Xianhai,Mandal, Mihirbaran,Zhao, Zhiqiang,Pissarnitski, Dmitri,Zhou, Wei,Aslanian, Robert,Zhu, Zhaoning,Greenlee, William,Clader, John,Zhang, Lili,Cohen-Williams, Mary,Jones, Nicholas,Hyde, Lynn,Palani, Anandan
scheme or table, p. 664 - 669 (2011/02/27)
We herein report the discovery of four series of fused 5,6-bicyclic heterocycles as γ-secretase modulators. Synthesis and SAR of these series are discussed. These compounds represent a new class of γ-secretase modulators that demonstrate moderate to good