116835-10-0Relevant academic research and scientific papers
Assembly of Diversely Substituted Quinolines via Aerobic Oxidative Aromatization from Simple Alcohols and Anilines
Li, Jixing,Zhang, Jinlong,Yang, Huameng,Jiang, Gaoxi
, p. 3284 - 3290 (2017)
An aerobic oxidative aromatization of simple aliphatic alcohols and anilines under the Pd(OAc)2/2,4,6-Collidine/Br?nsted acid catalytic system has been established, providing a direct approach for the preparation of diverse substituted quinoline derivatives in high yields with wide functional group tolerance. Practically, the protocol can be easily scaled up to gram-scale and was utilized in the concise formal synthesis of a promising herbicide candidate.
One-pot and convenient conversion of 5-azidopyrazole-4-carboxaldehyde to pyrazolo[3,4-b]pyridines
Zheng, Airong,Zhang, Wei,Pan, Jinhui
, p. 1549 - 1556 (2006)
A one-pot and convenient synthesis of multisubstituted pyrazolo[3, 4-b]pyridines in moderate to high yields has been achieved by a two-step reaction: diazo-transfer of 5-azido-1-phenylpyrazole-4-carboxaldehydes to ketones in ethanolic KOH to give 5-amino-
