1174985-52-4Relevant academic research and scientific papers
Discovery of novel arylpyrazole series as potent and selective opioid receptor-like 1 (ORL1) antagonists
Kobayashi, Kensuke,Uchiyama, Minaho,Ito, Hirokatsu,Takahashi, Hirobumi,Yoshizumi, Takashi,Sakoh, Hiroki,Nagatomi, Yasushi,Asai, Masanori,Miyazoe, Hiroshi,Tsujita, Tomohiro,Hirayama, Mioko,Ozaki, Satoshi,Tani, Takeshi,Ishii, Yasuyuki,Ohta, Hisashi,Okamoto, Osamu
scheme or table, p. 3627 - 3631 (2010/08/06)
The synthesis and biological evaluation of new potent opioid receptor-like 1 antagonists are presented. A structure-activity relationship (SAR) study of arylpyrazole lead compound 1 obtained from library screening identified compound 31, (1S,3R)-N-{[1-(3-
