1179538-82-9Relevant academic research and scientific papers
Synthesis of 3-acyl-2-arylindole via palladium-catalyzed isocyanide insertion and oxypalladation of alkyne
Nanjo, Takeshi,Yamamoto, Sho,Tsukano, Chihiro,Takemoto, Yoshiji
, p. 3754 - 3757 (2013/08/23)
The synthesis of 3-acyl-2-arylindole derivatives was performed through palladium-catalyzed isocyanide insertion and oxypalladation of an alkyne. As a result of the introduction of internal nucleophiles, domino cyclization was also achieved for the synthes
3-Aroylindoles via copper-catalyzed cyclization of N-(2-iodoaryl)enaminones
Bernini, Roberta,Cacchi, Sandro,Fabrizi, Giancarlo,Filisti, Eleonora,Sferrazza, Alessio
experimental part, p. 1480 - 1484 (2009/10/17)
3-Aroylindoles have been prepared via copper-catalyzed cyclization of N-(2-iodoaryl)enaminones, readily available from 2-iodoanilines and α,β-ynones. The reaction tolerates a variety of useful functionalities including ether, keto, cyano, bromo, and chlor
