1200442-82-5Relevant academic research and scientific papers
Displacement assay for the detection of stabilizers of inactive kinase conformations
Klüter, Sabine,Grütter, Christian,Naqvi, Tabassum,Rabiller, Matthias,Simard, Jeffrey R.,Pawar, Vijaykumar,Getlik, Matth?us,Rauh, Daniel
experimental part, p. 357 - 367 (2010/06/11)
Targeting protein kinases with small molecules outside the highly conserved ATP pocket to stabilize inactive kinase conformations is becoming a more desirable approach in kinase inhibitor research, since these molecules have advanced pharmacological prope
