1200442-83-6Relevant academic research and scientific papers
Displacement assay for the detection of stabilizers of inactive kinase conformations
Klüter, Sabine,Grütter, Christian,Naqvi, Tabassum,Rabiller, Matthias,Simard, Jeffrey R.,Pawar, Vijaykumar,Getlik, Matth?us,Rauh, Daniel
, p. 357 - 367 (2010)
Targeting protein kinases with small molecules outside the highly conserved ATP pocket to stabilize inactive kinase conformations is becoming a more desirable approach in kinase inhibitor research, since these molecules have advanced pharmacological prope
