1202802-49-0Relevant academic research and scientific papers
Design, synthesis, and biological evaluation of highly potent small molecule-peptide conjugates as new HIV-1 fusion inhibitors
Wang, Chao,Shi, Weiguo,Cai, Lifeng,Lu, Lu,Wang, Qian,Zhang, Tianhong,Li, Jinglai,Zhang, Zhenqing,Wang, Kun,Xu, Liang,Jiang, Xifeng,Jiang, Shibo,Liu, Keliang
, p. 2527 - 2539 (2013/05/21)
The small molecule fusion inhibitors N-(4-carboxy-3-hydroxyphenyl)-2,5- dimethylpyrrole (NB-2) and N-(3-carboxy-4-hydroxyphenyl)-2,5-dimethylpyrrole (A12) target a hydrophobic pocket of HIV-1 gp41 and have moderate anti-HIV-1 activity. In this
