120742-08-7Relevant articles and documents
Synthesis of the Novel ?-(Benzyloxymethyl)-Protected Histidine Analogue of Statine. Inhibition of Penicillopepsin by Pepstatin-Derived Peptides Containing Different Statine Side-Chain Derivatives
Maibaum, Juergen,Rich, Daniel H.
, p. 1571 - 1576 (2007/10/02)
The synthesis of aspartic proteinase inhibitors derived from a new histidine side-chain analogue of statine (Sta), (3S,4S)-4-amino-3-hydroxy-5-(imidazol-4-yl)pentanoic acid (HiSta, 20), is reported.Boc-HiSta(BOM)-OMe (7) was prepared in 16percent overall