122946-88-7Relevant articles and documents
Synthesis of Pyranoindoles as Conformationally Restricted Analogues of the Serotonin Antagonist ICS 205-930 and as Precursors to 2-Vinylindoles
Macor, John E.,Ryan, Kevin,Newman, Michael E.
, p. 4785 - 4795 (1989)
A useful synthesis of some pyranoindoles is described that allows access to conformationally restricted analogues of the serotonin (5HT3) antagonist, ICS 205-930.These pyranoindoles can be converted in one step to 2-vinylindole derivatives.