123213-67-2Relevant academic research and scientific papers
Thiophene systems. 12. Analogues of ketanserin and ritanserin as selective 5-HT2 antagonists
Press, JB,Russell, RK,McNally, JJ,Rampulla, RA,Falotico, R,et al.
, p. 807 - 813 (2007/10/02)
A series of thieno-, - and pyrimidinedione derivatives was prepared with N-3 substitution containing the side chains of ketanserin and ritanserin.The best of these thiophene analogues were the isosteres of ketanserin which were up to
THIENO-AND FUROPYRIMIDINE-2,4-DIONE PIPERIDINE DERIVATIVES AS SEROTONIN ANTAGONISTS AND ALPHA ADRENERGIC BLOCKING AGENTS
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, (2008/06/13)
Novel thienopyrimidine-2,4-dione piperidine derivatives and novel furo[3,4-d]pyrimidine-2,4-dione piperidine derivatives are described. The novel piperidine derivatives are selective serotonin antagonists and alpha adrenergic blocking agents with cardiova
