1235485-56-9Relevant academic research and scientific papers
A vHTS approach for the identification of β-adrenoceptor ligands
Tasler, Stefan,Baumgartner, Roland,Aschenbrenner, Andrea,Ammendola, Astrid,Wolf, Kristina,Wieber, Tanja,Schachtner, Josef,Blisse, Marcus,Quotschalla, Udo,Ney, Peter
, p. 3399 - 3404 (2010)
Using a vHTS based on a pharmacophore alignment on known β3-adrenoceptor ligands, a set of intriguing β-adrenoceptor ligands was identified, optimization of which resulted in a selective and potent human β2-AR antagonist.
