1240516-35-1Relevant articles and documents
Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigation
Procopiou, Panayiotis A.,Ford, Alison J.,Graves, Rebecca H.,Hall, David A.,Hodgson, Simon T.,Lacroix, Yannick M.L.,Needham, Deborah,Slack, Robert J.
, p. 2730 - 2733 (2012/05/31)
Synthesis and preliminary SAR of the N1 substituent of a novel series of indazole sulfonamide chemokine receptor 4 (CCR4) antagonist is reported. Compound 7r was identified for further development.
NOVEL COMPOUNDS
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Page/Page column 47, (2010/09/05)
Indazole compounds, processes for their preparation, intermediates usable in these processes, pharmaceutical compositions containing such compounds and their use in therapy.