124687-30-5Relevant articles and documents
Selective Inhibition of γ-Aminobutyric Acid Aminotransferase by (3R,4R),(3S,4S)- and (3R,4S),(3S,4R)-4-Amino-5-fluoro-3-phenylpentanoic Acids
Silverman, Richard B.,Nanavati, Shrenik M.
, p. 931 - 936 (2007/10/02)
(3R,4R),(2S,4S)- and (3R,4S),(3S,4R)-4-amino-5-fluoro-3-phenylpentanoic acid (1a and 1b) were synthesized and studied as selective inactivators of γ-aminobutyric acid (GABA) aminotransferase.Neither compound caused time-dependent inactivation of the enzym