1248-54-0Relevant academic research and scientific papers
Synthesis and structure–activity relationships of novel arylpiperazines as potent antagonists of α1-adrenoceptor
Silva, Renata Oliveira,de Oliveira, Andressa Souza,Nunes Lemes, Laís Flávia,de Camargo Nascente, Luciana,Coelho do Nascimento Nogueira, Patrícia,Silveira, Edilberto R.,Brand, Guilherme D.,Vistoli, Giulio,Cilia, Antonio,Poggesi, Elena,Buccioni, Michela,Marucci, Gabriella,Bolognesi, Maria Laura,Romeiro, Luiz Antonio Soares
, p. 601 - 610 (2016/07/22)
Arylpiperazines 2–11 were synthesized, and their biological profiles at α1-adrenergic receptors (α1-ARs) assessed by binding assays in CHO cells expressing human cloned subtypes and by functional experiments in isolated rat vas deferens (α1A), spleen (α1B
