1258977-03-5Relevant articles and documents
QUINAZOLINE BASED RESPIRATORY SYNCYTIAL VIRUS INHIBITORS
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, (2015/05/19)
Compounds of Formula (I), wherein R1, R2, R3, R4 and n are defined herein, are useful as inhibitors of RSV.
PYRROLIDINO HETEROCYCLES
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Page/Page column 45-46, (2014/01/07)
The invention relates to compounds of formula I wherein A1, A2, A3, B, R1, R2, R3 and R4 are as defined in the description and in the claims, as well as physiologically acceptable salts thereof. These compounds inhibit PDE10A and can be used as medicaments.
A General synthetic procedure for 2-chloromethyl-4(3H)-quinazolinone derivatives and their utilization in the preparation of novel anticancer agents with 4-anilinoquinazoline scaffolds
Li, Hong-Ze,He, Hai-Yun,Han, Yuan-Yuan,Gu, Xin,He, Lin,Qi, Qing-Rong,Zhao, Ying-Lan,Yang, Li
experimental part, p. 9473 - 9485 (2011/02/27)
In our ongoing research on novel anticancer agents with 4-anilinoquinazoline scaffolds, a series of novel 2-chloromethyl-4(3H)- quinazolinones were needed as key intermediates. An improved one-step synthesis of 2-chloromethyl-4(3H)-quinazolinones utilizin