1262328-71-1Relevant articles and documents
Identification of diaryl ether-based ligands for estrogen-related receptor α as potential antidiabetic agents
Patch, Raymond J.,Searle, Lily L.,Kim, Alexander J.,De, Debyendu,Zhu, Xizhen,Askari, Hossein B.,O'Neill, John C.,Abad, Marta C.,Rentzeperis, Dionisios,Liu, Jianying,Kemmerer, Michael,Lin, Ling,Kasturi, Jyotsna,Geisler, John G.,Lenhard, James M.,Player, Mark R.,Gaul, Micheal D.
experimental part, p. 788 - 808 (2011/04/22)
Estrogen-related receptor R (ERRR) is an orphan nuclear receptor that has been functionally implicated in the regulation of energy homeostasis. Herein is described the development of diaryl ether based thiazolidenediones, which function as selective ligan