1263324-74-8Relevant articles and documents
Regioselective synthesis of 1,3,5- and 1,3,4,5-substituted pyrazoles via acylation of N-Boc-N-substituted hydrazones
Tinarelli, Alessandro,Righi, Paolo,Rosini, Goffredo,Andreotti, Daniele,Profeta, Roberto,Spada, Simone
experimental part, p. 612 - 617 (2011/03/19)
Acylation of N-Boc-N-methylhydrazones followed by TFA treatment affords regioselective access to substituted pyrazoles. Both regioisomers of 1-methyl-3,5-disubstituted-1H-pyrazoles can be selectively obtained. This procedure can also be employed for the r