1268262-16-3Relevant academic research and scientific papers
Protein kinase affinity reagents based on a 5-aminoindazole scaffold
Krishnamurty, Ratika,Brock, Amanda M.,Maly, Dustin J.
supporting information; experimental part, p. 550 - 554 (2011/02/27)
Affinity reagents that target protein kinases are powerful tools for signal transduction research. Here, we describe a general set of kinase ligands based on a 5-aminoindazole scaffold. This scaffold can readily be derivatized with diverse binding elements and immobilized analogs allow selective enrichment of protein kinases from complex mixtures.
