1284288-91-0Relevant academic research and scientific papers
Solid-phase synthesis of skeletally diverse benzofused sultams via palladium-catalyzed cyclization
Chen, Wenteng,Li, Zhi,Ou, Lili,Giulianott, Marc A.,Houghten, Richard A.,Yu, Yongping
, p. 1456 - 1458 (2011)
The solid-phase synthesis of sultams from resin-bound amino acids is described. The sulfonylation of the resin-bound primary amines afforded the requisite secondary amines, after which the intramolecular Buchwald-Hartwig-type coupling forms the C-S bond.
