128830-76-2Relevant academic research and scientific papers
Novel Acyl-CoA:Cholesterol Acyltransferase Inhibitors. Synthesis and Biological Activity of 3-Quinolylurea Derivatives
Tawada, Hiroyuki,Harcourt, Myles,Kawamura, Noriaki,Kajino, Masahiro,Ishikawa, Eiichiro,et al.
, p. 2079 - 2084 (2007/10/02)
A series of 3-quinolylurea derivatives (1) was synthesized and evaluated for acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activity.For in vitro studies, the most potent inhibitory activity was found in derivatives having substituents at the 6,7-
Quinoline derivatives, their production and use
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, (2008/06/13)
Quinoline derivatives of the formula: STR1 , wherein R is hydrogen, alkyl or aralkyl; m and n are 0 or 1, and each of rings A, B and C can have substituents, which are useful as inhibitors for acyl-CoA:Cholesterolacyltransferase.
