1304141-60-3Relevant articles and documents
Chiral 2,3-disubstituted indolines from indoles and aldehydes by organocatalyzed tandem synthesis involving reduction by trichlorosilane
Chen, Lin,Wang, Chao,Zhou, Li,Sun, Jian
supporting information, p. 2224 - 2230 (2014/07/21)
The organocatalytic trichlorosilane reduction system has been successfully utilized to develop a multi-step tandem approach for the easy preparation of chiral 2-methyl-3-alkylindolines starting from simple 2-methylindoles and aldehydes. A broad range of c
Pd-Catalyzed asymmetric hydrogenation of 3-(toluenesulfonamidoalkyl)indoles
Duan, Ying,Chen, Mu-Wang,Chen, Qing-An,Yu, Chang-Bin,Zhou, Yong-Gui
, p. 1235 - 1238 (2012/03/07)
A series of 2-substituted 3-(toluenesulfonamidoalkyl)indoles was synthesized by application of (EtO)2POH or iodine as the catalyst, and was hydrogenated using chiral Pd catalyst, giving the 2,3-disubstituted indolines with up to 97% ee. The Royal Society of Chemistry 2012.