1310687-65-0Relevant articles and documents
The discovery of novel 8-azabicyclo[3.2.1]octan-3-yl)-3-(4-chlorophenyl) propanamides as vasopressin V1A receptor antagonists
Napier, Susan,Wishart, Grant,Arbuckle, William,Baker, James,Barn, David,Bingham, Matilda,Brown, Angus,Byford, Alan,Claxton, Chris,Craighead, Mark,Buchanan, Kirsteen,Fielding, Lee,Gibson, Lindsay,Goodwin, Richard,Goutcher, Susan,Irving, Nicholas,MacSweeney, Cliona,Milne, Rachel,Mort, Chris,Presland, Jeremy,Sloan, Hazel,Thomson, Fiona,Turnbull, Zara,Young, Trevor
, p. 3163 - 3167 (2011/06/24)
The discovery of a novel series of 8-azabicyclo[3.2.1]octan-3-yl)-3-(4- chlorophenyl) propanamide antagonists of the vasopressin V1A receptor is disclosed. Compounds 47 and 48 were found to be high affinity, selective vasopressin V1A antagonists.