1314582-27-8Relevant articles and documents
3-Acylindoles as versatile starting materials for pyridine ring annulation: Synthesis of 1-deazapurine isosteres
Knepper, Ingo,Iaroshenko, Viktor O.,Vilches-Herrera, Marcelo,Domke, Lutz,Mkrtchyan, Satenik,Zahid, Muhammad,Villinger, Alexander,Langer, Peter
experimental part, p. 5293 - 5303 (2011/08/04)
The reaction of electron-rich aminoheterocycles with 3-acyl- and 3-formylindoles results in indole ring opening and cyclocondensation to give heteroannulated pyridines, which can be regarded as purine isosteres. The transformations reported herein represe