1333309-66-2Relevant academic research and scientific papers
A highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine using a simple β-amino alcohol organocatalyst for a practical synthetic methodology of oseltamivir intermediate
Suttibut, Chonticha,Kohari, Yoshihito,Igarashi, Ko,Nakano, Hiroto,Hirama, Masafumi,Seki, Chigusa,Matsuyama, Haruo,Uwai, Koji,Takano, Nobuhiro,Okuyama, Yuko,Osone, Kenichi,Takeshita, Mitsuhiro,Kwon, Eunsang
supporting information; experimental part, p. 4745 - 4748 (2011/10/02)
An easily prepared chiral amino alcohol catalyst was found to provide an efficient synthetic intermediate of oseltamivir with excellent chemical yield and enantioselectivity (up to 98% yield and up to 98% ee) in enantioselective Diels-Alder reactions of 1
A novel chiral oxazolidine organocatalyst for the synthesis of an oseltamivir intermediate using a highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine
Nakano, Hiroto,Osone, Kenichi,Takeshita, Mitsuhiro,Kwon, Eunsang,Seki, Chigusa,Matsuyama, Haruo,Takano, Nobuhiro,Kohari, Yoshihito
supporting information; experimental part, p. 4827 - 4829 (2010/09/16)
Enantioselective Diels-Alder reactions of 1,2-dihydropyridines with acroleins using a novel chiral oxazolidine organocatalyst afforded chiral isoquinuclidines that is an efficient synthetic intermediate of oseltamivir, with fairly good chemical yield and
