1340595-72-3Relevant academic research and scientific papers
Novel diarylpyridinones, diarylpyridazinones and diarylphthalazinones as potential HIV-1 nonnucleoside reverse transcriptase inhibitors (NNRTIs)
Venkatraj, Muthusamy,Ari?n, Kevin K.,Heeres, Jan,Dirié, Bertrand,Joossens, Jurgen,Van Goethem, Sebastiaan,Van Der Veken, Pieter,Michiels, Johan,Vande Velde, Christophe M.L.,Vanham, Guido,Lewi, Paul J.,Augustyns, Koen
, p. 5924 - 5934 (2011/10/31)
In this Letter, we report on diarylpyridinone, diarylpyridazinone and diarylphthalazinone analogs as potential inhibitors of HIV-1 nonnucleoside reverse transcriptase (NNRTIs). The most promising compounds in these series are three diarylpyridazinones 25a
