134675-58-4Relevant academic research and scientific papers
Synthesis and Biological Activity of CCK Heptapeptide Analogues. Effects of Conformational Constraints and Standard Modifications on Receptor Subtype Selectivity, Functional Activity in Vitro, and Appetite Suppression in Vivo
Holladay, Mark W.,Bennett, Michael J.,Tufano, Michael D.,Lin, C. W.,Asin, Karen E.,et al.
, p. 2919 - 2928 (2007/10/02)
A series of modifications of the CCK7 analogue (des-NH2)Tyr(SO3-)-Nle-Gly-Trp-Nle-Asp-Phe-NH2 was prepared and tested for binding to guinea pig CCK-A and CCK-B receptors and in CCK-A-mediated functional assays.Selected analogues also were teste
