134953-66-5Relevant articles and documents
Electrophilic amination: First direct transfer of NHBoc with Li t-butyl-N-tosyloxycarbamate
Genet,Mallart,Greck,Piveteau
, p. 2359 - 2362 (1991)
Lithium t-butyl-N-tosyloxycarbamate (LiBTOC) has been found to be an electrophilic aminating reagent. This species reacts with organometallic reagents, ester enolates and α-cuprophosphonates to provide primary amines as well as α-aminocarboxylic and phosphonic esters in their N-(Boc) protected form. (35-80% isolated yields).