1353776-73-4Relevant academic research and scientific papers
Copper-catalyzed highly regioselective 2-aryloxylation of 2,x-dihalopyridines
Zhou, Qizhong,Zhang, Bin,Du, Tieqi,Gu, Haining,Ye, Yuyuan,Jiang, Huajiang,Chen, Rener
, p. 327 - 333 (2013/01/15)
2,x-Dihalopyridines reacted with phenols catalyzed by CuI/TMEDA in the presence of Cs2CO3 in DMSO at 110 °C under nitrogen atmosphere for 24 h to afford 2-aryloxypyridines in good to high yields except p-nitrophenol. To expand this methodology, a vanilloid receptor ligand used in treatments was prepared in good yield. This method has potential utility in the synthesis of pharmaceuticals, agrochemicals and even natural products.
AZETIDINE DERIVATIVES
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Paragraph 0565; 0566; 0567; 0568; 0569; 0570, (2013/06/28)
Azetidine derivatives of which the following is exemplary and their use in the treatment of obesity, diabetes or dyslipidemia.
NEW COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF
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Page/Page column 48, (2012/06/30)
The invention relates to new piperidine derivatives of the formula I to their use as medicaments, to methods for their therapeutic use and to pharmaceutical compositions containing them.
