13575-40-1Relevant articles and documents
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Okafor,C.O.
, p. 126 (1967)
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Identification of a urea bioisostere of a triazole oxytocin antagonist
Brown, Alan,Ellis, Dave,Wallace, Olga,Ralph, Michael
scheme or table, p. 1851 - 1853 (2010/07/06)
A series of azetidine ureas were investigated as potential bioisosteres of previously reported azetidinyltriazole oxytocin antagonists. Although potency was somewhat reduced in several close-in analogues, one compound, 9, was both a potent oxytocin antagonist and demonstrated significant selectivity over the closely related vasopressin V1A receptor.