1369231-52-6Relevant articles and documents
5-Aryl-4-carboxamide-1,3-oxazoles: Potent and selective GSK-3 inhibitors
Gentile, Gabriella,Merlo, Giancarlo,Pozzan, Alfonso,Bernasconi, Giovanni,Bax, Benjamin,Bamborough, Paul,Bridges, Angela,Carter, Paul,Neu, Margarete,Yao, Gang,Brough, Caroline,Cutler, Geoffrey,Coffin, Aaron,Belyanskaya, Svetlana
, p. 1989 - 1994 (2012/04/17)
5-Aryl-4-carboxamide-1,3-oxazoles are a novel, potent and selective series of GSK-3 inhibitors. The optimization of the series to yield compounds with cell activity and brain permeability is described.