1373162-46-9Relevant articles and documents
Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigation
Procopiou, Panayiotis A.,Ford, Alison J.,Graves, Rebecca H.,Hall, David A.,Hodgson, Simon T.,Lacroix, Yannick M.L.,Needham, Deborah,Slack, Robert J.
, p. 2730 - 2733 (2012/05/31)
Synthesis and preliminary SAR of the N1 substituent of a novel series of indazole sulfonamide chemokine receptor 4 (CCR4) antagonist is reported. Compound 7r was identified for further development.