137451-39-9Relevant academic research and scientific papers
Mild and general method for the synthesis of sulfonamides
Garcia Ruano, Jose Luis,Parra, Alejandro,Yuste, Francisco,Mastranzo, Virginia M.
, p. 311 - 319 (2008/12/22)
Reaction of methyl sulfinates with lithium amides followed by 3-chloroperoxybenzoic acid oxidation of the resulting sulfinamides provides primary, secondary, and tertiary alkane-, arene-and heteroarenesulfonamides in high yields. This constitutes a mild and facile experimental protocol that avoids the use of hazardous, unstable, or volatile reagents and does not affect the configurational stability of the amines. Georg Thieme Verlag Stuttgart.
Some Studies on Peptide Analogues Involving the Sulphinamide Group
Merricks, David,Sammes, Peter G.,Walker, Edward R. H.,Henrick, Kim,McPartlin, Mary M.
, p. 2169 - 2176 (2007/10/02)
The title compounds are of interest as possible transition state inhibitors of peptidases.A route to N-(alkylsulphinyl)amino acids is described.A method for generating α-benzamidosulphinamides is reported; a general route to such systems failed owing to t
