1377834-33-7Relevant academic research and scientific papers
Structure-activity relationship of selected polyphenol derivatives as inhibitors of Bax/Bcl-xL interaction
Vo, Duc Duy,Gautier, Fabien,Juin, Philippe,Grée, René
, p. 286 - 293 (2012/07/14)
This paper describes the synthesis of nine selected diaryl/heteroaryl- containing phenol and polyphenol derivatives which have been evaluated against Bax/Bcl-xL interaction in comparison with ABT-737. Using a BRET assay, six of these derivatives exhibit activity comparable to ABT-737 to disrupt Bax/Bcl-xL interaction. These preliminary results demonstrate that such polyphenol-derived molecules are attractive compounds regarding anticancer activity and that the phenol at position 3 is important regarding disruption of Bax/Bcl-xL interaction.
