1379604-20-2Relevant articles and documents
Stereoselective radiosynthesis of L- and D-3-[18F]fluoro-α-methyltyrosine
Castillo Meleán, Johnny,Humpert, Sven,Ermert, Johannes,Coenen, Heinz H.
, p. 202 - 207 (2015)
A three-step radiosynthesis is described which allows for the first time the preparation of L- and D-3-[18F]fluoro-α-methyltyrosine starting from [18F]fluoride. Corresponding 3-fluoro-4-formyl-benzylated Sch?llkopf derivatives were
1-[1-(BENZOYL)-PYRROLIDINE-2-CARBONYL]-PYRROLIDINE-2-CARBONITRILE DERIVATIVES
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Page/Page column 40, (2014/05/24)
The present invention relates to 1-[1-(benzoyl)-pyrrolidine-2-carbonyl]-pyrrolidine-2-carbonitrile derivatives having pharmacological activity formula (I) to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use in therapy and/or prophylaxis of a cognitive disorder.
4- (5-CYANO-PYRAZOL-1-YL) -PIPERIDINE DERIVATIVES AS GPR 119 MODULATORS
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Page/Page column 71, (2012/06/15)
Compounds that modulate the activity of the G-protein-coupled receptor GPR119 and their uses in the treatment of diseases linked to the modulation of the G-protein- coupled receptor GPR119 in animals are described herein.