1384067-04-2Relevant articles and documents
3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES
-
Page/Page column 68; 69, (2012/07/13)
The present invention relates to 3,8-diaza-bicyclo[4.2.0]oct-3-yl amide derivatives of formula (I), wherein the relative configuration of the diazabicyclooctane moiety is cis; and wherein Ar1, and Ar2 are as described in the description, to their preparation, to pharmaceutically acceptable salts thereof, and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and especially to their use as orexin receptor antagonists.