139403-39-7Relevant academic research and scientific papers
Synthesis, Structure, and Properties of New Lupinine O-Acyl Derivatives
Nurkenov,Nurmaganbetov, Zh. S.,Fazylov,Satpaeva, Zh. B.,Turdybekov,Seilkhanov,Talipov
, p. 506 - 508 (2019)
Acylation of the alkaloid lupinine produced O-cinnamoyllupinine and O-lipoyllupinine. The structure of O-cinnamoyllupinine was established by an X-ray crystal structure analysis.
SYNTHESIS AND ANTICHOLINESTERASE PROPERTIES OF NEW DERIVATIVES OF LUPININE AND EPILUPININE
Tlegenov, R. T.,Khaitbaev, Kh.,Tilyabaev, E.,Dalimov, D. N.,Abduvakhabov, A. A.,Uteniyazov, K. U.
, p. 55 - 57 (2007/10/02)
Esters of lupinine and epilupinine have been obtained by their acylation with isovaleroyl, cinnamoyl, trichloroacetyl, and trimethylacetyl chlorides.The methiodide derivatives of these esters have been investigated in reactions with the blood cholinesterase of warm-blooded animals.The interaction has a reversible nature, and the inhibition of the activity of the enzyme is both quantitative and qualitative in dependence on the structure of the acid taken and the conformational properties of the lupinine epimers.
