140677-17-4Relevant academic research and scientific papers
Synthesis of marine alkaloid: 8,9-Dihydrocoscinamide B and its analogues as Novel class of antileishmanial agents
Gupta, Leena,Talwar, Archna,Nishi,Palne, Shraddha,Gupta, Suman,Chauhan, Prem M.S.
, p. 4075 - 4079 (2008/02/08)
A series of marine alkaloid 8,9-dihydrocoscinamide B, its analogues and indolylglyoxylamide derivatives have been synthesized and screened for their in vitro antileishmanial activity profile in promastigote and amastigote models. Compounds 7 and 10 have shown 99-100% inhibition against promastigotes and 97-98% inhibition against amastigotes at a concentration of 10 μg/ml.
Benzodiazepine Receptor Affinity and Interaction of Some N-(Indol-3-ylglyoxylyl)amine Derivatives
Bianucci, Anna Maria,Settimo, Antonio Da,Settimo, Federico Da,Primofiore, Giampaolo,Martini, Claudia,et al.
, p. 2214 - 2220 (2007/10/02)
Several derivatives, in which tryptamine, tyramine, and dopamine moieties are linked to the indole nucleus by an oxalyl bridge, were tested for their ability to displace the specific binding of 3H>flunitrazepam from bovine brain membranes.GABA
