141075-56-1Relevant academic research and scientific papers
A short, stereospecific synthesis of dihydrooxazoles from serine and threonine derivatives
Wipf, Peter,Miller, Chris P.
, p. 907 - 910 (2007/10/02)
Cyclization of serine and threonine derivatives with Burgess reagent provides a one-step, streospecific access to 4,5-dihydrooxazoles. Noteworthy features of this new methodology include mild experimental conditions, and the absence of β-lactam, aziridine
AN INVESTIGATION OF THE MITSUNOBU REACTION IN THE PREPARATION OF PEPTIDE OXAZOLINES, THIAZOLINES, AND AZIRIDINES
Wipf, Peter,Miller, Chris P.
, p. 6267 - 6270 (2007/10/02)
The diisopropyl azodicarboxylate-triphenylphosphine mediated cyclization of serine and allo-threonine derivatives provides peptide oxazolines, whereas cyclization of threonine containing substrates leads to N-acyl aziridines.In the thiopeptide series, onl
