1416807-99-2

Upstream product

• 1416807-67-4 8-(2,6-diethyl-4-methylphenyl)-3-methoxytetrahydropyrazolo[1,2-a][1,2,5]triazepine-7,9-dione 
• 541-41-3 chloroformic acid ethyl ester 
• 1416808-55-3 C₂₁H₃₃N₃O₄ 
• 886230-70-2 (2,6-diethyl-4-methylphenyl)acetic acid chloride 

Relevant academic research and scientific papers

Herbicidal aryldiones incorporating a 5-methoxy-[1,2,5]triazepane ring

Novel 2-aryl-cyclic-1,3-diones containing a 5-methoxy-[1,2,5]triazepane unit were explored towards an effective and wheat safe control of grass weeds. Their preparation builds on the ease of synthetic access to 7-membered heterocyclic [1,2,5]triazepane building blocks. Substitution and pattern hopping in the phenyl moiety revealed structure–activity relationships in good agreement with previously disclosed observations amongst the pinoxaden family of acetyl-CoA carboxylase inhibitors. In light of basic physicochemical, enzyme inhibitory and binding site properties, the N-methoxy functionality effectively acts as a bioisostere of the ether group in the seven-membered hydrazine ring.

N-OXY PYRAZOLO-TRIAZEPINE-DIONE DERIVATIVES

Compounds of formula (I) wherein the substituents are as defined in claim 1, are useful as a pesticides and herbicides.