142003-47-2Relevant academic research and scientific papers
Design and Synthesis of Some Substrate Analogue Inhibitors of Phospholipase A2 and Investigations by NMR and Molecular Modeling into the Binding Interactions in the Enzyme-Inhibitor Complex
Bennion, Colin,Connolly, Stephen,Gensmantel, Nigel P.,Hallam, Catherine,Jackson, Clive G.,et al.
, p. 2939 - 2951 (1992)
A series of substrate analogue inhibitors of pancreatic phospholipase A2 has been designed and synthesized.The compounds were tested in a novel dual-screening system based on parallel assays with monomeric and micellar substrates.Intermolecular
