1420459-35-3Relevant academic research and scientific papers
Design, synthesis, and pharmacological characterization of N - And O-substituted 5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol analogues: Novel 5-HT2A/5-HT2C receptor agonists with pro-cognitive properties
Jensen, Anders A.,Plath, Niels,Pedersen, Martin H. F.,Isberg, Vignir,Krall, Jacob,Wellendorph, Petrine,Stensb?l, Tine B.,Gloriam, David E.,Krogsgaard-Larsen, Povl,Fr?lund, Bente
, p. 1211 - 1227 (2013/03/28)
The isoxazol-3-one tautomer of the bicyclic isoxazole, 5,6,7,8-tetrahydro- 4H-isoxazolo[4,5-d]azepin-3-ol (THAZ), has previously been shown to be a weak GABAA and glycine receptor antagonist. In the present study, the potential in this scaffold
