1427690-73-0Relevant articles and documents
Synthesis, biological evaluation, and molecular docking analysis of phenstatin based indole linked chalcones as anticancer agents and tubulin polymerization inhibitors
Kode, Jyoti,Kovvuri, Jeshma,Nagaraju, Burri,Jadhav, Shailesh,Barkume, Madan,Sen, Subrata,Kasinathan, Nirmal Kumar,Chaudhari, Pradip,Mohanty, Bhabani Shankar,Gour, Jitendra,Sigalapalli, Dilep Kumar,Ganesh Kumar,Pradhan, Trupti,Banerjee, Manisha,Kamal, Ahmed
supporting information, (2020/11/17)
A library of new phenstatin based indole linked chalcone compounds (9a-z and 9aa-ad) were designed and synthesized. Of these, compound 9a with 1-methyl, 2- and 3-methoxy substituents in the aromatic ring was efficacious against the human oral cancer cell
New (3-(1: H -benzo [d] imidazol-2-yl))/(3-(3 H -imidazo[4,5- b] pyridin-2-yl))-(1 H -indol-5-yl)(3,4,5-trimethoxyphenyl)methanone conjugates as tubulin polymerization inhibitors
Mullagiri, Kishore,Nayak, V. Lakshma,Sunkari, Satish,Mani, Geeta Sai,Guggilapu, Sravanthi Devi,Nagaraju, Burri,Alarifi, Abdullah,Kamal, Ahmed
supporting information, p. 275 - 281 (2018/03/08)
A series of new (3-(1H-benzo[d]imidazol-2-yl))/(3-(3H-imidazo[4,5-b]pyridin-2-yl))-(1H-indol-5-yl)(3,4,5-trimethoxyphenyl)methanone conjugates 4-6(a-i) were synthesized and evaluated for their antiproliferative activity on selected human cancer cell lines
Endowing indole-based tubulin inhibitors with an anchor for derivatization: Highly potent 3-substituted indolephenstatins and indoleisocombretastatins
álvarez, Raquel,Puebla, Pilar,Díaz, J. Fernando,Bento, Ana C.,García-Navas, Rósula,De La Iglesia-Vicente, Janis,Mollinedo, Faustino,Andreu, José Manuel,Medarde, Manuel,Peláez, Rafael
supporting information, p. 2813 - 2827 (2013/06/04)
Colchicine site ligands with indole B rings are potent tubulin polymerization inhibitors. Structural modifications at the indole 3-position of 1-methyl-5-indolyl-based isocombretastatins (1,1-diarylethenes) and phenstatins endowed them with anchors for fu
